Mostrati risultati da 1 a 50 di 140
Titolo Data di pubblicazione Autore(i) Rivista Editore
Valorization of Pistacia lentiscus L. Hydrodistillation By-Products: Phytochemical Profile and Multitarget Anti-Aging Activity of an Aqueous Extract 1-gen-2026 Fais, Antonella; Pintus, Francesca; Era, Benedetta; Floris, Sonia; Urru, Giulia; Sanjust, Enrico; Cocco, Emma; Maxia, Andrea; Masala, Valentina; Tuberoso, Carlo Ignazio Giovanni PLANTS -
2-Arylbenzofurans as Selective Cholinesterase Inhibitors: Design, Synthesis, and Evaluation as Alzheimer’s Disease Agents 1-gen-2026 Delogu, Giovanna Lucia; Begala, Michela; Novás, Manuel; João Matos, Maria; Piras, Franca; Floris, Sonia; Pintus, Francesca; Mancinelli, Michele; Era, Benedetta; Fais, Antonella BIOMOLECULES -
Investigating the Ligand-Binding Properties of N-arylbenzimidazoles as Novel Elastase Inhibitors 1-gen-2026 Pitasi, G.; Floris, S.; Mancuso, F.; Savoca, G.; Gitto, R.; Fais, A.; De Luca, L. CHEMMEDCHEM -
The Anti-Angiogenic Effect of Cynara cardunculus L. subsp. cardunculus Waste Product 1-gen-2025 Cacciola, Anna; D'Angelo, Valeria; De Gaetano, Federica; Fais, Antonella; Germanò, Maria Paola; Masala, Valentina; Olla, Stefania; Pistarà, Venerando; Stancanelli, Rosanna; Tuberoso, Carlo Ignazio Giovanni; Ventura, Cinzia Anna FOODS -
Inhibition of α-Glucosidase Activity and Islet Amyloid PolyPeptide Fibril Formation by Rubus ulmifolius Fruit Extract: A Potential Therapeutic Approach for Type 2 Diabetes Mellitus 1-gen-2025 Floris, Sonia; Noli, Barbara; Cocco, Cristina; Fais, Antonella; Era, Benedetta; Tuberoso, Carlo Ignazio Giovanni; Masala, Valentina; Piras, Franca; Sogos, Valeria; Di Petrillo, Amalia; De Agostini, Antonio; Pintus, Francesca; Sanna, Cinzia PLANTS -
Structure-based design and evaluation of tyrosinase inhibitors targeting both human and mushroom isozymes 1-gen-2025 Mirabile, S.; Pitasi, G.; Floris, S.; Schira, K.; Khettabi, L.; Soler-Lopez, M.; Scheuermann, J.; Gitto, R.; Germano, M. P.; Fais, A.; De Luca, L. RSC MEDICINAL CHEMISTRY -
Fatty acid profile and biological activity of supercritical fluid extract of Rosa canina L. seeds 1-gen-2025 Ibba, A.; Rosa, A.; Fais, A.; Era, B.; Porcedda, S.; Piras, A. NATURAL PRODUCT RESEARCH -
Aqueous Extract of Rubus ulmifolius Schott (Rosaceae) against Pathogenic Gram-Positive Oral Bacteria: an in Vitro Evaluation 1-gen-2025 Ibba, A.; Piras, A.; Era, B.; Fais, A.; Maxia, A.; Fais, S.; Orru, G.; Porcedda, S. LETTERS IN APPLIED NANOBIOSCIENCE -
Sustainable Synthesis of 1,2-Disubstituted Benzimidazoles as Promising α-Glucosidase Inhibitors: In Vitro and In Silico Evaluation 1-gen-2025 Tocco, Graziella; Laus, Antonio; Manis, Cristina; Caboni, Pierluigi; Fais, Antonella; Era, Benedetta PHARMACEUTICALS -
Xanthine Oxidase-Dependent Activation of NLPR3 Inflammasome in Epithelial Cells Sustains Inflammation in Inflammatory Bowel Disease 1-gen-2025 Di Petrillo, Amalia; Fais, Antonella; Raho, Nicola; Era, Benedetta; Cannea, Faustina Barbara; Padiglia, Alessandra; Grecu, Eleonora; Murtas, Daniela; Maxia, Cristina; Sogos, Valeria; Porcedda, Clara; Caboni, Pierluigi; Demurtas, Mauro; Favale, Agnese; Onali, Sara; Fantini, Massimo Claudio INFLAMMATORY BOWEL DISEASES -
Supercritical extraction from Rosa canina L. fruits: fatty acids composition and biological activities 1-gen-2024 Ibba, A.; Rosa, A.; Fais, A.; Era, B.; Porcedda, S.; Piras, A. LA RIVISTA ITALIANA DELLE SOSTANZE GRASSE -
Phytochemical Composition and Biological Activity 1-gen-2024 Fais, A.; Era, B. PLANTS -
Exploring the 1-(4-Nitrophenyl)-3-arylprop-2-en-1-one Scaffold for the Selective Inhibition of Monoamine Oxidase B 1-gen-2024 Meleddu, Rita; Fais, Antonella; Era, Benedetta; Floris, Sonia; Distinto, Simona; Lupia, Antonio; Cottiglia, Filippo; Onali, Alessia; Sanna, Erica; Secci, Daniela; Atzeni, Giulia; Demuru, Laura; Caboni, Pierluigi; Valenti, Donatella; Maccioni, Elias ACS MEDICINAL CHEMISTRY LETTERS -
Advances in Sardinian Withania somnifera (L.) Dunal crops through phytochemical and biological approaches 1-gen-2024 Maccioni, Delia; Falconieri, Danilo; Acquas, Elio; Kasture, Sanjay Bhaskar; Era, Benedetta; Fais, Antonella; Cocco, Emma; Maxia, Andrea INDUSTRIAL CROPS AND PRODUCTS -
Exploring Asphodelus microcarpus as a source of xanthine oxidase inhibitors: Insights from in silico and in vitro studies 1-gen-2024 DI PETRILLO, Amalia; Siguri, Chiara; Delogu, Giovanna L.; Fais, Antonella; Era, Benedetta; Floris, Sonia; Pintus, Francesca; Kumar, Amit; Fantini, MASSIMO CLAUDIO; Olla, Stefania CHEMICO-BIOLOGICAL INTERACTIONS -
Design, Synthesis, Structural Insights, Tyrosinase Inhibition, and Sun Protection Factor of New Thiosemicarbazone Derivatives 1-gen-2024 Masuri, Sebastiano; Era, Benedetta; Pintus, Francesca; Floris, Sonia; Meloni, Francesca; Pettinau, Francesca; Podda, Enrico; Cabiddu, MARIA GRAZIA; Fais, Antonella; Pivetta, Tiziana MOLECULES -
A New Class of Benzo[b]thiophene-chalcones as Cholinesterase Inhibitors: Synthesis, Biological Evaluation, Molecular Docking and ADME Studies 1-gen-2024 Delogu, GIOVANNA LUCIA; Begala, Michela; João Matos, Maria; Crucitti, Davide; Sogos, Valeria; Era, Benedetta; Fais, Antonella MOLECULES -
Computational Approach to Identifying New Chemical Entities as Elastase Inhibitors with Potential Antiaging Effects 1-gen-2024 Pitasi, G.; Brancale, A.; Floris, S.; Fais, A.; Gitto, R.; De Luca, L. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES -
Biological Potential of Asphodelus microcarpus Extracts: α-Glucosidase and Antibiofilm Activities In Vitro 1-gen-2024 Floris, S.; Pintus, F.; Fais, A.; Era, B.; Raho, N.; Siguri, C.; Orru, G.; Fais, S.; Tuberoso, C. I. G.; Olla, S.; Di Petrillo, A. MOLECULES -
Template Entrance Channel as Possible Allosteric Inhibition and Resistance Site for Quinolines Tricyclic Derivatives in RNA Dependent RNA Polymerase of Bovine Viral Diarrhea Virus 1-gen-2023 Srivastava, M.; Mittal, L.; Sarmadhikari, D.; Singh, V. K.; Fais, A.; Kumar, A.; Asthana, S. PHARMACEUTICALS -
Comparison of Different Green Extraction Techniques Used for the Extraction of Targeted Flavonoids from Edible Feijoa (Acca sellowiana (O.Berg) Burret) Flowers 1-gen-2023 Gil, Katarzyna Angelika; Jokić, Stela; Cikoš, Ana-Marija; Banožić, Marija; Jakovljević Kovač, Martina; Fais, Antonella; Tuberoso, Carlo Ignazio Giovanni PLANTS -
Phytochemicals in structure-based drug discovery 1-gen-2023 Kumar, A.; Baranwal, J.; Di Petrillo, A.; Floris, S.; Barse, B.; Fais, A. - Elsevier
Inhibitory Effect of Quercetin on Oxidative Endogen Enzymes: A Focus on Putative Binding Modes 1-gen-2023 Olla, S.; Siguri, C.; Fais, A.; Era, B.; Fantini, M. C.; Di Petrillo, A. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES -
Promising inhibition of diabetes-related enzymes and antioxidant properties of Ptilostemon casabonae leaves extract 1-gen-2023 Sanna, Cinzia; Fais, Antonella; Era, Benedetta; Delogu, Giovanna L; Sanna, Enrico; Dazzi, Laura; Rosa, Antonella; Marengo, Arianna; Rubiolo, Patrizia; De Agostini, Antonio; Floris, Sonia; Pintus, Francesca JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Hydroxylated Coumarin-Based Thiosemicarbazones as Dual Antityrosinase and Antioxidant Agents 1-gen-2023 Masuri, Sebastiano; Era, Benedetta; Pintus, Francesca; Cadoni, Enzo; Cabiddu, Maria Grazia; Fais, Antonella; Pivetta, Tiziana INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES -
Design of 3-Phenylcoumarins and 3-Thienylcoumarins as Potent Xanthine Oxidase Inhibitors: Synthesis, Biological Evaluation, and Docking Studies 1-gen-2023 Fais, A.; Pintus, F.; Era, B.; Floris, S.; Kumar, A.; Sarmadhikari, D.; Sogos, V.; Uriarte, E.; Asthana, S.; Matos, M. J. CHEMMEDCHEM -
Euphorbia characias Extract: Inhibition of Skin Aging-Related Enzymes and Nanoformulation 1-gen-2022 Pintus, F.; Floris, S.; Fais, A.; Era, B.; Porcedda, C.; Tuberoso, C. I. G.; Caddeo, C. PLANTS -
Quercetin and its derivates as antiviral potentials: A comprehensive review 1-gen-2022 Di Petrillo, A.; Orru, G.; Fais, A.; Fantini, M. C. PHYTOTHERAPY RESEARCH -
Biopolymer: a sustainable material for food and medical applications 1-gen-2022 Baranwal, Jaya; Barse, Brajesh; Fais, Antonella; Delogu, GIOVANNA LUCIA; Kumar, Amit POLYMERS -
Hydroxy-3-Phenylcoumarins as Multitarget Compounds for Skin Aging Diseases: Synthesis, Molecular Docking and Tyrosinase, Elastase, Collagenase and Hyaluronidase Inhibition, and Sun Protection Factor 1-gen-2022 Pintus, Francesca; Floris, Sonia; Fais, Antonella; Era, Benedetta; Kumar, Amit; Gatto, Gianluca; Uriarte, Eugenio; Matos, Maria João MOLECULES -
Design, Synthesis, and in Vitro Evaluation of 4-(4-Hydroxyphenyl)piperazine-Based Compounds Targeting Tyrosinase 1-gen-2022 Mirabile, Salvatore; Paola Germanò, Maria; Fais, Antonella; Lombardo, Lisa; Ricci, Federico; Floris, Sonia; Cacciola, Anna; Rapisarda, Antonio; Gitto, Rosaria; Laura De Luca, And CHEMMEDCHEM -
Supercritical extraction of volatile and fixed oils from Petroselinum crispum L. seeds: chemical composition and biological activity 1-gen-2022 Piras, A.; Porcedda, S.; Falconieri, D.; Fais, A.; Era, B.; Carta, G.; Rosa, A. NATURAL PRODUCT RESEARCH -
Structural insight of new butyrylcholinesterase inhibitors based on benzylbenzofuran scaffold 1-gen-2022 Delogu, Giovanna L.; Fais, Antonella; Pintus, Francesca; Goyal, Chinmayi; Matos, Maria J.; Era, Benedetta; Kumar, Amit PHARMACEUTICALS -
Structural Characterisation and Assessment of the Novel Bacillus amyloliquefaciens RK3 Exopolysaccharide on the Improvement of Cognitive Function in Alzheimer’s Disease Mice 1-gen-2021 Gangalla, Ravi; Gattu, Sampath; Palaniappan, Sivasankar; Ahamed, Maqusood; Macha, Baswaraju; Thampu, Raja Komuraiah; Fais, Antonella; Cincotti, Alberto; Gatto, Gianluca; Dama, Murali; Kumar, Amit POLYMERS -
Euphorbia characias: Phytochemistry and Biological Activities 1-gen-2021 Fais, Antonella; Delogu, Giovanna Lucia; Floris, Sonia; Era, Benedetta; Medda, Rosaria; Pintus, Francesca PLANTS -
Evaluation of novel 4-(4-fluorobenzyl)piperazin-1-yl]-based compounds as competitive tyrosinase inhibitors endowed with anti-melanogenic effects 1-gen-2021 Mirabile, Salvatore; Vittorio, Serena; Germanò, Maria Paola; Adornato, Ilenia; Ielo, Laura; Rapisarda, Antonio; Gitto, Rosaria; Pintus, Francesca; De Luca, Laura; Fais, Antonella CHEMMEDCHEM -
Washingtonia filifera seed extracts inhibit the islet amyloid polypeptide fibrils formations and α-amylase and α-glucosidase activity 1-gen-2021 Floris, S.; Fais, A.; Medda, R.; Pintus, F.; Piras, A.; Kumar, A.; Kus, P. M.; Westermark, G. T.; Era, B. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
A new biological prospective for the 2-phenylbenzofurans as inhibitors of α-glucosidase and of the islet amyloid polypeptide formation 1-gen-2021 Delogu, GIOVANNA LUCIA; Era, Benedetta; Floris, Sonia; Medda, Rosaria; Sogos, Valeria; Pintus, Francesca; Gatto, Gianluca; Kumar, Amit; Torstensdotter Westermark, Gunilla; Fais, Antonella INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES -
Anti-aging potential of extracts from Washingtonia filifera seeds 1-gen-2021 Era, B.; Floris, S.; Sogos, V.; Porcedda, C.; Piras, A.; Medda, R.; Fais, A.; Pintus, F. PLANTS -
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety 1-gen-2020 De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R. BIOORGANIC & MEDICINAL CHEMISTRY -
Substitution Effects on the Optoelectronic Properties of Coumarin Derivatives 1-gen-2020 Kumar, Amit; Baccoli, Roberto; Fais, Antonella; Cincotti, Alberto; Pilia, Luca; Gatto, Gianluca APPLIED SCIENCES -
Looking for new xanthine oxidase inhibitors: 3-Phenylcoumarins versus 2-phenylbenzofurans 1-gen-2020 Era, Benedetta; Delogu, Giovanna L.; Pintus, Francesca; Fais, Antonella; Gatto, Gianluca; Uriarte, Eugenio; Borges, Fernanda; Kumar, Amit; Matos, Maria J. INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES -
4-Fluorobenzylpiperazine-containing derivatives as efficient inhibitors of mushroom tyrosinase 1-gen-2020 Vittorio, Serena; Ielo, Laura; Mirabile, Salvatore; Gitto, Rosaria; Fais, Antonella; Floris, Sonia; Rapisarda, Antonio; Paola Germanò, Maria; De Luca, Laura CHEMMEDCHEM -
Supercritical CO2 Extraction of Waste Citrus Seeds: Chemical Composition, Nutritional and Biological Properties of Edible Fixed Oils 1-gen-2019 Rosa, Antonella; Era, Benedetta; Masala, Carla; Nieddu, Mariella; Scano, Paola; Fais, Antonella; Porcedda, Silvia; Piras, Alessandra EUROPEAN JOURNAL OF LIPID SCIENCE AND TECHNOLOGY -
Chemical composition and enzyme inhibition of Phytolacca dioica L. seeds extracts 1-gen-2019 DI PETRILLO, Amalia; María González-Paramás, Ana; Rosa, Antonella; Ruggiero, Valeria; Boylan, Fabio; Kumar, Amit; Pintus, Francesca; Santos-Buelga, Celestino; Fais, Antonella; Era, Benedetta JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
Phytochemical composition and the cholinesterase and xanthine oxidase inhibitory properties of seed extracts from the Washingtonia filifera palm fruit. 1-gen-2019 Floris, Sonia; Fais, Antonella; Rosa, Antonella; Piras, Alessandra; Marzouki, Hanen; Medda, Rosaria; Gonz´alez-Paramas, Ana M.; Kumar, Amit; Santos-Buelga, Celestino; Era, Benedetta RSC ADVANCES -
Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile 1-gen-2019 Ielo, L.; Deri, B.; Germanò, M. P.; Vittorio, S.; Mirabile, S.; Gitto, R.; Rapisarda, A.; Ronsisvalle, S.; Floris, S.; Pazy, Y.; Fais, A.; Fishman, A.; De, Luca EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY -
Synthesis, molecular docking and cholinesterase inhibitory activity of hydroxylated 2-phenylbenzofuran derivatives 1-gen-2019 Fais, Antonella; Kumar, Amit; Medda, Rosaria; Pintus, Francesca; Delogu, Francesco; Matos, Maria J.; Era, Benedetta; Delogu, Giovanna L. BIOORGANIC CHEMISTRY -
Antibacterial Activity and Molecular Docking Studies of a Selected Series of Hydroxy-3-arylcoumarins 1-gen-2019 Pisano, M. B.; Kumar, A.; Medda, R.; Gatto, G.; Pal, Rajesh; Fais, A.; Era, B.; Cosentino, S.; Uriarte, E.; Santana, L.; Pintus, F.; Matos, M. J. MOLECULES -
Evaluation of antioxidant activities and chemical composition of Washingtonia filifera extracts. 1-gen-2018 Floris, S.; Era, B.; Fais, A.; Porcedda, S.; Falconieri, D.; Rosa, A.; Marzouki, H.; Santos Buelga, C.; Piras, A. - -
Mostrati risultati da 1 a 50 di 140
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