Università degli Studi di Cagliari
Luca Didaci
Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential
2026-01-01 Saravanan, Venkatesan; Angeli, Andrea; Melfi, Francesco; Amodio, Nicola; Valentino, Ilenia; Gentile, Massimo; D'Agostino, Ilaria; Muthukumaradoss, Kathiravan; Zengin, Gokhan; Moi, Davide; Simsek, Rahime; Supuran, Claudiu T.; Carradori, Simone
Prokineticin 2 regulates the electrophysiological activity of gonadotropin-releasing hormone neurons via direct signalling in adult female mice
2026-01-01 Farkas, Imre; Göblyös, Barbara; Moi, Davide; Onnis, Valentina; Kalló, Imre; Liposits, Zsolt
Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity
2026-01-01 Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina
Anticancer potential of chalcones
2026-01-01 Moi, Davide; Onnis, Valentina; Deplano, Alberto
Chalcones. From Drug Discovery to Pharmaceutical Applications
2026-01-01 Carradori, Simone; Moi, Davide; D’Agostino, Ilaria
Catalytic Enantioselective Synthesis of Conformationally Stable C(sp2)−C(sp3) Naphthocoumarin Atropisomers
2026-01-01 Cabua, M. Chiara; Moi, Davide; Cocco, Emanuele; Onnis, Valentina; Podda, Enrico; Aitken, David J.; Carlone, Armando; Luisi, Renzo; Tuveri, Enrica; Parsons, Drew F.; Secci, Francesco
The prokineticin system and glia cells as pharmacological targets to control neuroinflammation and to relieve pain in a murine model of Fabry–Anderson disease
2026-01-01 Galimberti, Giulia; Franchi, Silvia; Amodeo, Giada; Romualdi, Patrizia; Candeletti, Sanzio; Rullo, Laura; Losapio, Loredana Maria; Onnis, Valentina; Moi, Davide; Riboldi, Benedetta; Magni, Giulia; Ceruti, Stefania; Sacerdote, Paola
Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides
2025-01-01 Moi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025-01-01 Citarella, Andrea; Belluti, Silvia; Bonanni, Davide; Moi, Davide; Piccinini, Isabella; Rinaldi, Arianna; Papulino, Chiara; Benedetti, Rosaria; Cuoghi, Laura; Ciolo, Stefano Di; Silvani, Alessandra; Altucci, Lucia; Pinzi, Luca; Franchini, Silvia; Passarella, Daniele; Sorbi, Claudia; Giannini, Clelia; Imbriano, Carol; Rastelli, Giulio
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025-01-01 Citarella, Andrea; Sibille, Giulia; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Col, Lorenzo Dal; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Gribaudo, Giorgio; Passarella, Daniele
Low‐Impact Synthesis of γ‐Lactones through Photoinduced Baeyer‐Villiger Oxidation of Cyclic Ketones
2024-01-01 Cabua, Maria Chiara; Velichko, Viktoria; Pilia, Luca; Moi, Davide; Secci, Francesco
Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors
2024-01-01 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina
Exploring the Antiviral Potential of Esters of Cinnamic Acids with Quercetin
2024-01-01 Manca, Valeria; Chianese, Annalisa; Palmas, Vanessa; Etzi, Federica; Zannella, Carla; Moi, Davide; Secci, Francesco; Serreli, Gabriele; Sarais, Giorgia; Morone, Maria Vittoria; Galdiero, Massimiliano; Onnis, Valentina; Manzin, Aldo; Sanna, Giuseppina
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024-01-01 Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele
Two-step continuous flow-driven synthesis of 1,1-cyclopropane aminoketones
2024-01-01 Velichko, Viktoria; Moi, Davide; Soddu, Francesco; Scipione, Roberto; Podda, Enrico; Luridiana, Alberto; Cambie, Dario; Secci, Francesco; Cabua, Maria Chiara
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro
2023-01-01 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors
2023-01-01 Moi, Davide; Vittorio, Serena; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Synthesis of SARS-CoV-2 Mpro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses
2023-01-01 Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Dimasi, Alessandro; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives
2023-01-01 Citarella, Andrea; Dimasi, Alessandro; Moi, Davide; Passarella, Daniele; Scala, Angela; Piperno, Anna; Micale, Nicola
Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity
2023-01-01 Moi, Davide; Deplano, Alessandro; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer
2023-01-01 Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio
Dual Targeting Strategies on Histone Deacetylase 6 (HDAC6) and Heat Shock Protein 90 (Hsp90)
2022-01-01 Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio
Synthesis of potent and selective HDAC6 inhibitors led to unexpected opening of a quinazoline ring
2022-01-01 Moi, Davide; Citarella, Andrea; Bonanni, Davide; Pinzi, Luca; Passarella, Daniele; Silvani, Alessandra; Giannini, Clelia; Rastelli, Giulio
Continuous-Flow Synthesis of Arylthio-Cyclopropyl Carbonyl Compounds
2022-01-01 Moi, Davide; Cabua, Maria Chiara; Velichko, Viktoria; Cocco, Andrea; Chiappone, Annalisa; Mocci, Rita; Porcu, Stefania; Piras, Monica; Bianco, Stefano; Pesciaioli, Fabio; Secci, Francesco
Synthesis and Antiproliferative Effect of Halogenated Coumarin Derivatives
2022-01-01 Dettori, Tinuccia; Sanna, Giuseppina; Cocco, Andrea; Serreli, Gabriele; Deiana, Monica; Palmas, Vanessa; Onnis, Valentina; Pilia, Luca; Melis, Nicola; Moi, Davide; Caria, Paola; Secci, Francesco
Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications
2021-01-01 Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bonanni, Davide; Rastelli, Giulio
Inhibitors of histone deacetylase 6 based on a novel 3-hydroxy-isoxazole zinc binding group
2021-01-01 Linciano, Pasquale; Pinzi, Luca; Belluti, Silvia; Chianese, Ugo; Benedetti, Rosaria; Moi, Davide; Altucci, Lucia; Franchini, Silvia; Imbriano, Carol; Sorbi, Claudia; Rastelli, Giulio
Monopharmacology, polypharmacology and PROTAC approaches in drug discovery: investigation of enzyme inhibitors and antioxidant compounds
2020-02-06
Synthesis and evaluation of antioxidant and antiproliferative activity of 2-arylbenzimidazoles
2020-01-01 Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors
2020-01-01 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Piras, Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
In-Vitro Evaluation of Antioxidant, Antiproliferative and Photo-Protective Activities of Benzimidazolehydrazone Derivatives
2020-01-01 Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2020-01-01 Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors
2019-01-01 Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gianfranco; Onnis, Valentina; Potter, Barry V. L.
Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones
2019-01-01 Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation
2019-01-01 Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina
Selective Inhibition of Histone Deacetylase 10: Hydrogen Bonding to the Gatekeeper Residue is Implicated
2019-01-01 Géraldy, Magalie; Morgen, Michael; Sehr, Peter; Steimbach, Raphael; Moi, Davide; Ridinger, Johannes; Oehme, Ina; Witt, Olaf; Malz, Mona; Nogueira, Mauro S; Koch, Oliver; Gunkel, Nikolas; Miller, Aubry K
Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity
2018-01-01 Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina
Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy
2018-01-01 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T.
Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2018-01-01 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T.
| Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
|---|---|---|---|---|
| Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential | 1-gen-2026 | Saravanan, Venkatesan; Angeli, Andrea; Melfi, Francesco; Amodio, Nicola; Valentino, Ilenia; Gentile, Massimo; D'Agostino, Ilaria; Muthukumaradoss, Kathiravan; Zengin, Gokhan; Moi, Davide; Simsek, Rahime; Supuran, Claudiu T.; Carradori, Simone | PHARMACEUTICALS | - |
| Prokineticin 2 regulates the electrophysiological activity of gonadotropin-releasing hormone neurons via direct signalling in adult female mice | 1-gen-2026 | Farkas, Imre; Göblyös, Barbara; Moi, Davide; Onnis, Valentina; Kalló, Imre; Liposits, Zsolt | FRONTIERS IN ENDOCRINOLOGY | - |
| Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity | 1-gen-2026 | Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina | PHARMACEUTICALS | - |
| Anticancer potential of chalcones | 1-gen-2026 | Moi, Davide; Onnis, Valentina; Deplano, Alberto | - | Elsevier |
| Chalcones. From Drug Discovery to Pharmaceutical Applications | 1-gen-2026 | Carradori, Simone; Moi, Davide; D’Agostino, Ilaria | - | Elsevier |
| Catalytic Enantioselective Synthesis of Conformationally Stable C(sp2)−C(sp3) Naphthocoumarin Atropisomers | 1-gen-2026 | Cabua, M. Chiara; Moi, Davide; Cocco, Emanuele; Onnis, Valentina; Podda, Enrico; Aitken, David J.; Carlone, Armando; Luisi, Renzo; Tuveri, Enrica; Parsons, Drew F.; Secci, Francesco | ADVANCED SYNTHESIS & CATALYSIS | - |
| The prokineticin system and glia cells as pharmacological targets to control neuroinflammation and to relieve pain in a murine model of Fabry–Anderson disease | 1-gen-2026 | Galimberti, Giulia; Franchi, Silvia; Amodeo, Giada; Romualdi, Patrizia; Candeletti, Sanzio; Rullo, Laura; Losapio, Loredana Maria; Onnis, Valentina; Moi, Davide; Riboldi, Benedetta; Magni, Giulia; Ceruti, Stefania; Sacerdote, Paola | PAIN | - |
| Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides | 1-gen-2025 | Moi, Davide; Carradori, Simone; Gallorini, Marialucia; Mencarelli, Noemi; Deplano, Alberto; Angeli, Andrea; Vittorio, Serena; Supuran, Claudiu T.; Onnis, Valentina | PHARMACEUTICALS | - |
| Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer | 1-gen-2025 | Citarella, Andrea; Belluti, Silvia; Bonanni, Davide; Moi, Davide; Piccinini, Isabella; Rinaldi, Arianna; Papulino, Chiara; Benedetti, Rosaria; Cuoghi, Laura; Ciolo, Stefano Di; Silvani, Alessandra; Altucci, Lucia; Pinzi, Luca; Franchini, Silvia; Passarella, Daniele; Sorbi, Claudia; Giannini, Clelia; Imbriano, Carol; Rastelli, Giulio | JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity | 1-gen-2025 | Citarella, Andrea; Sibille, Giulia; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Col, Lorenzo Dal; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Gribaudo, Giorgio; Passarella, Daniele | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Low‐Impact Synthesis of γ‐Lactones through Photoinduced Baeyer‐Villiger Oxidation of Cyclic Ketones | 1-gen-2024 | Cabua, Maria Chiara; Velichko, Viktoria; Pilia, Luca; Moi, Davide; Secci, Francesco | EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | - |
| Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors | 1-gen-2024 | Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T.; Onnis, Valentina | ACS MEDICINAL CHEMISTRY LETTERS | - |
| Exploring the Antiviral Potential of Esters of Cinnamic Acids with Quercetin | 1-gen-2024 | Manca, Valeria; Chianese, Annalisa; Palmas, Vanessa; Etzi, Federica; Zannella, Carla; Moi, Davide; Secci, Francesco; Serreli, Gabriele; Sarais, Giorgia; Morone, Maria Vittoria; Galdiero, Massimiliano; Onnis, Valentina; Manzin, Aldo; Sanna, Giuseppina | VIRUSES | - |
| Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells | 1-gen-2024 | Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Two-step continuous flow-driven synthesis of 1,1-cyclopropane aminoketones | 1-gen-2024 | Velichko, Viktoria; Moi, Davide; Soddu, Francesco; Scipione, Roberto; Podda, Enrico; Luridiana, Alberto; Cambie, Dario; Secci, Francesco; Cabua, Maria Chiara | CHEMICAL COMMUNICATIONS | - |
| Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro | 1-gen-2023 | Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia | MOLECULES | - |
| Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors | 1-gen-2023 | Moi, Davide; Vittorio, Serena; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | MOLECULES | - |
| Synthesis of SARS-CoV-2 Mpro inhibitors bearing a cinnamic ester warhead with in vitro activity against human coronaviruses | 1-gen-2023 | Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Dimasi, Alessandro; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele | ORGANIC & BIOMOLECULAR CHEMISTRY | - |
| Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives | 1-gen-2023 | Citarella, Andrea; Dimasi, Alessandro; Moi, Davide; Passarella, Daniele; Scala, Angela; Piperno, Anna; Micale, Nicola | BIOMOLECULES | - |
| Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity | 1-gen-2023 | Moi, Davide; Deplano, Alessandro; Angeli, Andrea; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | MOLECULES | - |
| Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer | 1-gen-2023 | Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Dual Targeting Strategies on Histone Deacetylase 6 (HDAC6) and Heat Shock Protein 90 (Hsp90) | 1-gen-2022 | Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio | CURRENT MEDICINAL CHEMISTRY | - |
| Synthesis of potent and selective HDAC6 inhibitors led to unexpected opening of a quinazoline ring | 1-gen-2022 | Moi, Davide; Citarella, Andrea; Bonanni, Davide; Pinzi, Luca; Passarella, Daniele; Silvani, Alessandra; Giannini, Clelia; Rastelli, Giulio | RSC ADVANCES | - |
| Continuous-Flow Synthesis of Arylthio-Cyclopropyl Carbonyl Compounds | 1-gen-2022 | Moi, Davide; Cabua, Maria Chiara; Velichko, Viktoria; Cocco, Andrea; Chiappone, Annalisa; Mocci, Rita; Porcu, Stefania; Piras, Monica; Bianco, Stefano; Pesciaioli, Fabio; Secci, Francesco | MOLECULES | - |
| Synthesis and Antiproliferative Effect of Halogenated Coumarin Derivatives | 1-gen-2022 | Dettori, Tinuccia; Sanna, Giuseppina; Cocco, Andrea; Serreli, Gabriele; Deiana, Monica; Palmas, Vanessa; Onnis, Valentina; Pilia, Luca; Melis, Nicola; Moi, Davide; Caria, Paola; Secci, Francesco | MOLECULES | - |
| Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications | 1-gen-2021 | Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bonanni, Davide; Rastelli, Giulio | ACS OMEGA | - |
| Inhibitors of histone deacetylase 6 based on a novel 3-hydroxy-isoxazole zinc binding group | 1-gen-2021 | Linciano, Pasquale; Pinzi, Luca; Belluti, Silvia; Chianese, Ugo; Benedetti, Rosaria; Moi, Davide; Altucci, Lucia; Franchini, Silvia; Imbriano, Carol; Sorbi, Claudia; Rastelli, Giulio | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Monopharmacology, polypharmacology and PROTAC approaches in drug discovery: investigation of enzyme inhibitors and antioxidant compounds | 6-feb-2020 | - | - | Università degli Studi di Cagliari |
| Synthesis and evaluation of antioxidant and antiproliferative activity of 2-arylbenzimidazoles | 1-gen-2020 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | BIOORGANIC CHEMISTRY | - |
| Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors | 1-gen-2020 | Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Piras, Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | BIOORGANIC CHEMISTRY | - |
| In-Vitro Evaluation of Antioxidant, Antiproliferative and Photo-Protective Activities of Benzimidazolehydrazone Derivatives | 1-gen-2020 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | PHARMACEUTICALS | - |
| Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 1-gen-2020 | Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; Alothman, Zeid A.; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors | 1-gen-2019 | Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gianfranco; Onnis, Valentina; Potter, Barry V. L. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones | 1-gen-2019 | Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | BIOORGANIC CHEMISTRY | - |
| Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation | 1-gen-2019 | Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Selective Inhibition of Histone Deacetylase 10: Hydrogen Bonding to the Gatekeeper Residue is Implicated | 1-gen-2019 | Géraldy, Magalie; Morgen, Michael; Sehr, Peter; Steimbach, Raphael; Moi, Davide; Ridinger, Johannes; Oehme, Ina; Witt, Olaf; Malz, Mona; Nogueira, Mauro S; Koch, Oliver; Gunkel, Nikolas; Miller, Aubry K | JOURNAL OF MEDICINAL CHEMISTRY | - |
| Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity | 1-gen-2018 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy | 1-gen-2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T. | BIOORGANIC CHEMISTRY | - |
| Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 1-gen-2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T. | BIOORGANIC CHEMISTRY | - |
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